| 1BAK |
|
SIGNAL TRANSDUCTION PLECKSTRIN HOMOLOGY DOMAIN OF G-PROTEIN COUPLED RECEPTOR KINASE 2 (BETA-ADRENERGIC RECEPTOR KINASE 1), C-TERMINAL EXTENDED, NMR, 20 STRUCTURES |
| 3CIK |
2.75 |
Human GRK2 in Complex with Gbetagamma subunits |
| 3KRW |
2.9 |
Human GRK2 in complex with Gbetgamma subunits and balanol (soak) |
| 3KRX |
3.1 |
Human GRK2 in complex with Gbetgamma subunits and balanol (co-crystal) |
| 3V5W |
2.07 |
Human G Protein-Coupled Receptor Kinase 2 in Complex with Soluble Gbetagamma Subunits and Paroxetine |
| 4MK0 |
2.4 |
Crystal structure of G protein-coupled receptor kinase 2 in complex with a a rationally designed paroxetine derivative |
| 4PNK |
2.56 |
G protein-coupled receptor kinase 2 in complex with GSK180736A |
| 5HE1 |
3.15 |
Human GRK2 in complex with Gbetagamma subunits and CCG224062 |
| 5UKK |
2.6 |
Human GRK2 in complex with human G-beta-gamma subunits and CCG211998 (14ak) |
| 5UKL |
2.15 |
Human GRK2 in complex with Gbetagamma subunits and CCG222886 (14bd) |
| 5UUU |
2.7 |
Design, Synthesis, and Evaluation of the First Selective and Potent G-protein-Coupled Receptor Kinase 2 (GRK2) Inhibitor for the Potential Treatment of Heart Failure |
| 5UVC |
2.65 |
Design, Synthesis, and Evaluation of the First Selective and Potent G-protein-Coupled Receptor Kinase 2 (GRK2) Inhibitor for the Potential Treatment of Heart Failure |
| 5WG3 |
2.896 |
Human GRK2 in complex with Gbetagamma subunits and CCG258748 |
| 5WG4 |
2.31 |
Human GRK2 in complex with Gbetagamma subunits and CCG257284 |
| 5WG5 |
3.1 |
Human GRK2 in complex with Gbetagamma subunits and CCG224061 |
| 6C2Y |
2.74 |
Human GRK2 in complex with Gbetagamma subunits and CCG257142 |
| 6U7C |
2.44 |
Human GRK2 in complex with Gbetagamma subunits and CCG258747 |
| 7K7L |
2.539 |
Structure of a hit for G Protein Coupled Receptor Kinase 2 (GRK2) Inhibitor for the Potential Treatment of Heart Failure |
| 7K7Z |
2.60609 |
Structure of a hit for G Protein Coupled Receptor Kinase 2 (GRK2) Inhibitor for the Potential Treatment of Heart Failure |
| 7PWD |
2.6 |
Structure of an inhibited GRK2-G-beta and G-gamma complex |
