| 2O8J |
1.8 |
Human euchromatic histone methyltransferase 2 |
| 3DM1 |
2.4 |
Crystal structure of the complex of human chromobox homolog 3 (CBX3) with peptide |
| 3K5K |
1.7 |
Discovery of a 2,4-Diamino-7-aminoalkoxy-quinazoline as a Potent Inhibitor of Histone Lysine Methyltransferase, G9a |
| 3RJW |
2.56 |
Crystal structure of histone lysine methyltransferase g9a with an inhibitor |
| 4NVQ |
2.03 |
Human G9a in Complex with Inhibitor A-366 |
| 5JHN |
1.67 |
Structure of G9a SET-domain with Histone H3K9Ala mutant peptide and bound S-adenosylmethionine |
| 5JIN |
1.85 |
Structure of G9a SET-domain with Histone H3K9M mutant peptide and bound S-adenosylmethionine |
| 5JIY |
1.48 |
Structure of G9a SET-domain with Histone H3K9norLeucine mutant peptide and bound S-adenosylmethionine |
| 5JJ0 |
1.72 |
Structure of G9a SET-domain with Histone H3K9M peptide and excess SAH |
| 5T0K |
1.7 |
Structure of G9a SET-domain with H3K9M mutant peptide and SAM |
| 5T0M |
1.896 |
A histone H3K9M mutation traps histone methyltransferase Clr4 to prevent heterochromatin spreading |
| 5TTF |
1.72 |
Crystal structure of catalytic domain of G9a with MS012 |
| 5TUY |
2.6 |
Structure of human G9a SET-domain (EHMT2) in complex with inhibitor MS0124 |
| 5V9I |
1.74 |
Crystal structure of catalytic domain of G9a with MS0105 |
| 5VSC |
1.4 |
Structure of human G9a SET-domain (EHMT2) in complex with inhibitor 13 |
| 5VSE |
1.6 |
Structure of human G9a SET-domain (EHMT2) in complex with inhibitor 17: N~2~-cyclopentyl-6,7-dimethoxy-N~2~-methyl-N~4~-(1-methylpiperidin-4-yl)quinazoline-2,4-diamine |
| 6MM1 |
1.9 |
Structure of the cysteine-rich region from human EHMT2 |
| 7BTV |
2.0 |
Crystal structure of EHMT2 SET domain in complex with compound 5. |
| 7BUC |
2.6 |
Crystal structure of EHMT2 SET domain in complex with compound 13 |
| 7DCF |
1.8 |
Crystal structure of EHMT2 SET domain in complex with compound 10 |
| 7T7L |
2.2 |
Structure of human G9a SET-domain (EHMT2) in complex with covalent inhibitor (Compound 1) |
| 7X73 |
1.49 |
Structure of G9a in complex with RK-701 |
| 7XUA |
1.87 |
Structure of G9a in complex with compound 10a |
| 7XUB |
2.0 |
Structure of G9a in complex with compound 10d |
| 7XUC |
1.67 |
Structure of G9a in complex with compound 11a |
| 7XUD |
1.45 |
Structure of G9a in complex with compound 26a |
